Synthesis and biological evaluation of new Benzimidazole derivatives
نویسندگان
چکیده
منابع مشابه
Synthesis and Anticandidal Activity Evaluation of New Benzimidazole-Thiazole Derivatives.
Azole-based antifungal agents constitute one of the important classes of antifungal drugs. Hence, in the present work, 12 new benzimidazole-thiazole derivatives 3a-3l were synthesized to evaluate their anticandidal activity against C.albicans, C.glabrata, C.krusei, and C.parapsilopsis. The structures of the newly synthesized compounds 3a-3l were confirmed by IR, ¹H-NMR, 13C-NMR, and ESI-MS spec...
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Aseries of piperidine derivatives was synthesis by the reaction between substituted benzaldhyde ,pentanone-3,and ammonium acetate by refluxining for 1-2 hr in ethanol and the derivatives refluxed with (4,4'-Diaminodiphenyl sulphone) yielded bispiperidine ,the structures of the synthesized compounds were confirmed by spectroscopy analysis , The reported compounds were screened for their antibact...
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ژورنال
عنوان ژورنال: Al-Mustansiriyah Journal of Science
سال: 2018
ISSN: 2521-3520,1814-635X
DOI: 10.23851/mjs.v29i1.127